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Search Results for " h1 receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
T7477 Antazoline Others
Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.
T36949 Niaprazine 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff...
T9353 OXOMEMAZINE AChR , Histamine Receptor
Oxomemazine is a phenothiazine-based histamine H1-receptor blocker with pronounced antimuscarinic activity. Oxomemazine is a selective antagonist of mycotoxins M1 receptors, showing high (Ki=84 nM, M1 receptors) and low ...
T1278 Astemizole Laridal,Histaminos,Paralergin Potassium Channel , Histamine Receptor
Astemizole (Laridal) is a synthetic piperidinyl-benzimidazol derivative with antiallergic properties, acts as a reversible competitive inhibitor of histamine H1 receptors, with less anticholinergic effects compared to re...
TN1008 Psoralenoside CaMK , Calcium Channel , Histamine Receptor
Psoralenoside is a natural product isolated from the fruits of Psoralea corylifolia, shows estrogen-like activity, osteoblastic proliferation accelerating activity, antitumor effects and antibacterial activity.
T0147 Clemastine fumarate HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate) Autophagy , Histamine Receptor
Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.
T13352 Wy 49051 Wy-49051 Histamine Receptor
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
T6405 Bepotastine Besilate Talion,TAU 284,Bepreve,Bepotastine Beslilate Histamine Receptor
Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
T0118 Mizolastine SL 850324 Histamine Receptor
Mizolastine (SL 850324) (IC50= 47 nM) is a histamine H1-receptor antagonist.It is used in the treatment of allergic reactions such as hay fever (seasonal allergic rhinitis), hives.
T13566 Bamirastine TAK-427 Histamine Receptor
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on allergic skin inflammation.
T2533 Alcaftadine R89674,Lastacaft Histamine Receptor
Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
T4250 Bilastine Bilaxten Histamine Receptor
Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of action.
T3979 Emedastine LY188695,Emadine Histamine Receptor
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blocks histamine by binding to H1 receptors, thus blocking its...
T2200 Hydroxyzine dihydrochloride Hydroxyzine 2HCl Histamine Receptor
Hydroxyzine dihydrochloride (Hydroxyzine 2HCl) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIR...
T22354 Levocetirizine Dihydrochloride Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride Histamine Receptor
Levocetirizine Dihydrochloride (Xyzal Dihydrochloride) is a third-generation peripheral H1-receptor antagonist. Acting as an antihistaminic agent, it specifically targets the histamine H1-receptor. Levocetirizine Dihydro...
T16778 Rocastine AHR-11325 Histamine Receptor
Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
T22501 2-Pyridylethylamine dihydrochloride Histamine Receptor
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
T22713 Decloxizine Histamine Receptor
Decloxizine is a H1 receptor antagonist
T0263 Chloropyramine hydrochloride Nilfan,Alergosan,Halopyramine hydrochloride FAK , VEGFR , Histamine Receptor
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
T7085 Mebhydrolin Mebhydroline Histamine Receptor
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.

Compounds

Antazoline
T7477
Synonym:
Target: Others
Niaprazine
T36949
Synonym:
Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
OXOMEMAZINE
T9353
Synonym:
Target: AChR, Histamine Receptor
Astemizole
T1278
Synonym: Laridal,Histaminos,Paralergin
Target: Potassium Channel, Histamine Receptor
Psoralenoside
TN1008
Synonym:
Target: CaMK, Calcium Channel, Histamine Receptor
Clemastine fumarate
T0147
Synonym: HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate)
Target: Autophagy, Histamine Receptor
Wy 49051
T13352
Synonym: Wy-49051
Target: Histamine Receptor
Bepotastine Besilate
T6405
Synonym: Talion,TAU 284,Bepreve,Bepotastine Beslilate
Target: Histamine Receptor
Mizolastine
T0118
Synonym: SL 850324
Target: Histamine Receptor
Bamirastine
T13566
Synonym: TAK-427
Target: Histamine Receptor
Alcaftadine
T2533
Synonym: R89674,Lastacaft
Target: Histamine Receptor
Bilastine
T4250
Synonym: Bilaxten
Target: Histamine Receptor
Emedastine
T3979
Synonym: LY188695,Emadine
Target: Histamine Receptor
Hydroxyzine dihydrochloride
T2200
Synonym: Hydroxyzine 2HCl
Target: Histamine Receptor
Levocetirizine Dihydrochloride
T22354
Synonym: Xyzal Dihydrochloride,(-)-Cetirizine Dihydrochloride
Target: Histamine Receptor
Rocastine
T16778
Synonym: AHR-11325
Target: Histamine Receptor
2-Pyridylethylamine dihydrochloride
T22501
Synonym:
Target: Histamine Receptor
Decloxizine
T22713
Synonym:
Target: Histamine Receptor
Chloropyramine hydrochloride
T0263
Synonym: Nilfan,Alergosan,Halopyramine hydrochloride
Target: FAK, VEGFR, Histamine Receptor
Mebhydrolin
T7085
Synonym: Mebhydroline
Target: Histamine Receptor
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TargetMol